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Details on Person UniProt:Q12774 ARHGEF5

Class:IdReferenceGeneProduct:50261
_chainChangeLogchain:1-1597 added on Fri February 6 2015
_displayNameUniProt:Q12774 ARHGEF5
_timestamp2024-11-03 19:49:57
chainchain:1-1597
checksum93EC1B1D7E1198C5
commentFUNCTION Guanine nucleotide exchange factor which activates Rho GTPases (PubMed:15601624). Strongly activates RHOA (PubMed:15601624). Also strongly activates RHOB, weakly activates RHOC and RHOG and shows no effect on RHOD, RHOV, RHOQ or RAC1 (By similarity). Involved in regulation of cell shape and actin cytoskeletal organization (PubMed:15601624). Plays a role in actin organization by generating a loss of actin stress fibers and the formation of membrane ruffles and filopodia (PubMed:14662653). Required for SRC-induced podosome formation (By similarity). Involved in positive regulation of immature dendritic cell migration (By similarity).SUBUNIT Interacts with SRC (By similarity). Forms a ternary complex with SRC and the PI3K 85 kDa subunit (By similarity). Interacts with and is activated by the heterodimer formed by GNB1 and GNG2 (By similarity). Interacts with ODAM (via C-terminus) (PubMed:25911094). Interacts with RHOA (By similarity).INTERACTION A number of additional isoforms are detected in primary breast tumors but not in normal tissues.TISSUE SPECIFICITY Ubiquitously expressed with highest levels in placenta. High levels are also found in colon, kidney, trachea, prostate, liver, pancreas, pituitary gland, thyroid gland and mammary gland. In fetal tissues, expressed at high levels in kidney, lung and liver (PubMed:15601624). Expressed at low levels in lung and heart (PubMed:14662653).DOMAIN The PH domain binds to phosphoinositides and is essential for podosome formation.PTM Activation of SRC induces tyrosine phosphorylation of ARHGEF5.SEQUENCE CAUTION Extended N-terminus.
descriptionrecommendedName: Rho guanine nucleotide exchange factor 5 alternativeName: Ephexin-3 alternativeName: Guanine nucleotide regulatory protein TIM alternativeName: Oncogene TIM alternativeName: Transforming immortalized mammary oncogene alternativeName: p60 TIM
geneNameARHGEF5
TIM
identifierQ12774
isSequenceChangedFALSE
keywordAlternative splicing
Cell junction
Cell projection
Cytoplasm
Guanine-nucleotide releasing factor
Lipid-binding
Methylation
Nucleus
Phosphoprotein
Proteomics identification
Proto-oncogene
Reference proteome
SH3 domain
modified[InstanceEdit:9836292] Weiser, Joel, 2023-05-25
[InstanceEdit:9852000] Weiser, Joel, 2023-11-03
[InstanceEdit:9926675] Weiser, Joel, 2024-11-03
nameARHGEF5
referenceDatabase[ReferenceDatabase:2] UniProt
referenceGene[ReferenceDNASequence:8991720] ENSEMBL:ENSG00000050327 ARHGEF5 [Homo sapiens]
secondaryIdentifierARHG5_HUMAN
A6NNJ2
Q6ZML7
sequenceLength1597
species[Species:48887] Homo sapiens
(isoformParent)[ReferenceIsoform:384459] UniProt:Q12774-2 ARHGEF5 [Homo sapiens]
[ReferenceIsoform:405517] UniProt:Q12774-1 ARHGEF5 [Homo sapiens]
(referenceEntity)[EntityWithAccessionedSequence:8873909] ARHGEF5 [cytosol] [Homo sapiens]
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No pathways have been reviewed or authored by UniProt:Q12774 ARHGEF5 (50261)